李杰 - 18新利体育

李杰

  姓名：李杰
  职称：教授

  部门：化学学院
  联系方式：

Email: jjackli@suda.edu.cn

01. 2020- 至今教授，18新利体育 ‒材料与化学化工学部，苏州，江苏

10. 2017- 11. 2019 慕尼黑大学‒化学与药学院博士后研究员，慕尼黑，德国； (合作导师：Prof. Dr. Paul Knochel)

10. 2015- 10. 2017 特聘研究员，江南大学‒药学院, 无锡，江苏

08. 2015- 10. 2015 访问学者，中国医学科学院药物研究所‒药物化学室(肖志艳研究员)

11. 2011- 07. 2015 哥廷根大学‒有机化学与分子生物化学系博士，哥廷根，德国；(博士学位‒“summa cum laude”; 合作导师：Prof. Dr. Lutz Ackermann).

08. 2009- 10. 2011 中国医学科学院药物研究所‒药物化学室(硕士交换生；导师：肖志艳研究员).

09. 2008- 07. 2009 沈阳药科大学‒(天然)药物化学系硕士(导师：华会明教授).

09. 2004- 06. 2008 (学士学位). 天津商业大学‒制药工程系

学历及学术经历: 2012年至今以一作或通讯作者在J. Am. Chem. Soc., Angew. Chem. Int. Ed., ACS Catal., Org. Lett., Adv. Synth. Catal., Chem. Eur. J., J. Org. Chem.,等期刊上发表学术论文20余篇；入选2016年江苏省双创人才；目前完成国家自然科学基金青年项目一项、江苏省自然科学基金青年基金一项。

研究领域：金属有机化学 & 药物化学

代表性论文（*通讯作者）：

1. Z. Zhang, L. Liu, Y. Wang, Y. Zhang,J. Li*, Electrophilic Amination with Anthranils through Cobalt(III)-Catalyzed C(sp³)‒H Activation.Synthesis 2020,DOI: 10.1055/s-0039-1690087.

2. J. Li*, Q. Ren, X. Cheng, K. Karaghiosoff, P. Knochel*, Chromium(II)-Catalyzed Diastereoselective and Chemoselective Csp²‒Csp³ Cross-Couplings Using Organomagnesium Reagents. J. Am. Chem. Soc.2019, 141, 18127‒18135.

3. S. Han, S. Liu, L. Liu, L. Ackermann, J. Li*, Cobalt-Catalyzed Diastereoselective Difluoroalkyaltion/Giese Addition Domino Reactions. Org. Lett.2019, 21, 5387‒5391. (Front Cover)

4. J. Li*, P. Knochel*, Chromium-Catalyzed Cross-Couplings and Related Reactions. Synthesis2019, 51, 2100‒2106.

5. J. Li*, E. Tan, N. Keller, Y.-H. Chen, P. M. Zehetmaier, A. C. Jakowetz, T. Bein*, P. Knochel*, Cobalt-Catalyzed Electrophilic Amination with Anthranils: An Expedient Route to Condensed Quinolines. J. Am. Chem. Soc.2019, 141, 98‒103. (highlighted inSynfact2019)

6. M. Tang, Y. Li, S. Han, L. Liu, L. Ackermann, J. Li*, Rhodium(III)-Catalyzed C‒H Alkylation/Nucleophilic Addition Domino Reaction. Eur. J. Org. Chem. 2019, 660‒664.

7. Y. Da, S. Han, X. Du, S. Liu, L. Liu, J. Li*, Copper(I)-Catalyzed Oxydifluoroalkylation of Alkenes: A Route to Functionalization Lactones. Org. Lett. 2018, 20. 5149‒5152.

8. J. Li, P. Knochel*, Cobalt-Catalyzed Cross-Couplings between Alkenyl Acetates and Aryl or Alkenyl Zinc Pivalates. Angew. Chem. Int. Ed. 2018, 57, 11436‒11440.

9. Liang-Hua Zou*, Cong Zhao, Ping-Gui Li, Ying Wang, J. Li*, Transition-Metal-Free C−S Bond Formation: Synthesis of Polysubstituted Diaryl Sulfides and α‑Thioarylcarbonyl Compounds. J. Org. Chem. 2017, 82, 12892–12898.

10. X. Zhang*, H. Zheng, J. Li*, F. Xu, J. Zhao, H. Yan*, Selective Catalytic B–H Arylation of o-Carboranyl Aldehydes by a Transient Directing Strategy. J. Am. Chem. Soc. 2017, 139, 14511‒14517.

11. Z. Zhang, S. Han, M. Tang, L. Ackermann*, J. Li*, C–H Alkylations of (Hetero)Arenes by Maleimides and Maleate Ester through Versatile Cobalt(III) Catalysis.Org. Lett. 2017, 19, 3135–3318.

12. S. Han, W. Ma, Z. Zhang, L. Liu, M. Tang, J. Li*, Mild C(sp³)‒H Alkylation of 8-Methylquinolines with α,β-Unsaturated Carbonyl Compounds by Rhodium(III) Catalysis.Asain J.Org. Chem. 2017, 6, 1014‒1018.(Front Cover)

13. J. Li*, Z. Zhang, W. Ma, M. Tang, D. Wang, L.-H. Zou, Mild Cobalt(III)-Catalyzed C‒H Hydroarylation of Conjugated C＝C/C＝O Bonds. Adv. Synth. Catal. 2017, 359,1717–1724.

14. M. Moselage^†, J. Li^†(Co-first author), F. Kramm, L. Ackermann*, Ruthenium(II)-Catalyzed Decarbamoylative C–C Arylations and Alkylations. Angew. Chem. Int. Ed. 2017, 55, 5341–5344.

15. Z. Zhang, M. Tang, S. Han, L. Ackermann, J. Li*, Carboxylate Enhanced Rhodium(III)-Catalyzed Aryl C–H Alkylation with Conjugated Alkenes under Mild Conditions.J. Org. Chem. 2017, 82, 664–672.

16. W. Ma*, P. Gandeepan*, J. Li, L. Ackermann*, Recent Advances in Positional-Selective Alkenylations: Removable Guidance for Twofold C‒H Activation. Org. Chem. Front. 2017, 4, 1435‒1467.

17. Z. Zhang, M. Tang, L. Zang, L.-H. Zou, J. Li*, Thermolysis of 2-Diazo-3-aryl ketoesters: New Route to α-Aryl Malonates and Aromatic Esters. Tetrahedron Lett. 2016, 57, 5681–5684.

18. J. Li*, Z. Zhang, M. Tang, X. Zhang, J. Jin, Selective Synthesis of Isoquinolines by Rhodium(III)-Catalyzed C–H/N–H Functionalization with α-Substituted Ketones. Org. Lett. 2016, 18, 3898–3901.

19. J. Li*, M. Tang, L. Zang, X. Zhang, Z. Zhang, L. Ackermann*, Amidines for Versatile Cobalt(III)-Catalyzed Synthesis of Isoquinolines through C–H Functionalization with Diazo Compounds. Org. Lett. 2016, 18, 2742–2745. (highlighted inOrganic Chemistry Portal2017)

20. M. Moselage^†, J. Li^†(Co-first author), L. Ackermann*, Cobalt-Catalyzed C–H Activation. ACS Catal. 2016, 6, 498–525.

21. J. Li, L. Ackermann*, Cobalt(III)-Catalyzed Aryl and Alkenyl C–H Aminocarbonylation with Isocyanates and Acyl Azides. Angew. Chem. Int. Ed. 2015, 54, 8551–8554.

22. J. Li, L. Ackermann*, Cobalt-Catalyzed C–H Cyanation of Arenes and Heteroarenes. Angew. Chem. Int. Ed. 2015, 54, 3635–3638. (Selected as hot paper, highlighted inChemCatChem 2015, 7, 732).

23. J. Li, L. Ackermann*, Cobalt-Catalyzed C–H Arylations with Weakly-Coordinating Amindes and Tetrazoles: Expedient Route to Angiotensin-II-Receptor Blockers. Chem. Eur. J. 2015, 21, 5718–5722.

24. J. Li, L. Ackermann*, Carboxylate-Assisted Ruthenium(II)-Catalyzed C–H Activations of Monodentate Amides with Conjugated Alkenes. Org. Chem. Front. 2015, 2, 1035–1039.

25. J. Li, M. John, L. Ackermann*, Amidines for Versatile Ruthenium(II)-Catalyzed Oxidative C–H Activations with Internal Alkynes and Acrylates. Chem. Eur. J. 2014, 20, 5403–5408.

26. J. Li, L. Ackermann*, Ruthenium-Catalyzed Oxidative Alkyne Annulation by C–H Activation on Ketimines. Tetrahedron 2014, 70, 3342–3348.

27. J. Li, H.-M. Hua, Y-B. Tang, S. Zhang, E. Ohkoshi, K.-H Lee, Z. Xiao*, Synthesis and Evaluation of Novel Podophyllotoxin Analogs. Bioorg. Med. Chem. Lett. 2012, 22, 4293–4295.